Concurrent Post
-
Faculty of Science and Engineering Graduate School of Advanced Science and Engineering
Details of a Researcher
Updated on 2022/05/26
Faculty of Science and Engineering Graduate School of Advanced Science and Engineering
理工学術院総合研究所 兼任研究員
University of Tokyo Graduate School, Division of Pharmaceutical Sciences
University of Tokyo Graduate School, Division of Pharmaceutical Sciences
University of Tokyo Faculty of Pharmaceutical Science
東京大学 博士(薬学)
Ph.D.
博士(薬学)
国際複素環化学会
アメリカ化学会
International Heterocyclic Chemistry
American Chemical Society
有機合成化学協会
日本薬学会
日本化学会
Synthetic organic chemistry
Bioorganic chemistry
Structural organic chemistry and physical organic chemistry
Pharmaceutical chemistry and drug development sciences
Chemical Pharmacology,Molecular Pharmacology
Research on Au(I)-catalyzed ene-yne cycloisomerization for construction of quassinoid scaffold
Yuta Oki, Masahisa Nakada
Tetrahedron Letters 59 ( 10 ) 926 - 929 2018.03
Substituent effect on the reaction pathway of Au(I)-catalyzed ene-yne cycloisomerization
Yuta Oki, Masahisa Nakada
Tetrahedron Letters 59 ( 10 ) 922 - 925 2018.03
Research on Liebeskind-Srogl coupling/intramolecular Diels-Alder reaction cascade
Tomohiro Fujii, Yuta Oki, Masahisa Nakada
Tetrahedron Letters 59 ( 10 ) 882 - 886 2018.03
Synthesis and Reaction of ortho-Benzoquinone Monohemiaminals
Emi Saito, Yuri Matsumoto, Akihiko Nakamura, Yuki Namera, Masahisa Nakada
Organic Letters 20 ( 3 ) 692 - 695 2018.02
Catalytic Asymmetric Intramolecular Cyclopropanation of alpha-Diazo-alpha-Silyl Acetate
Saori Inoue, Kotaro Nagatani, Haruka Tezuka, Yunosuke Hoshino, Masahisa Nakada
SYNLETT 28 ( 9 ) 1065 - 1070 2017.06 [Refereed]
Enantio- and Stereoselective Construction of Atisane Scaffold via Organocatalytic Intramolecular Michael Reaction and Diels-Alder Reaction
Hiroko Sekita, Kyohei Adachi, Ippei Kobayashi, Yusuke Sato, Masahisa Nakada
ORGANIC LETTERS 19 ( 9 ) 2390 - 2393 2017.05 [Refereed]
Enantioselective preparation of C-ring fragment of cotylenin A via catalytic asymmetric intramolecular cyclopropanation of alpha-diazo beta-keto ester
Kotaro Nagatani, Yunosuke Hoshino, Haruka Tezuka, Masahisa Nakada
TETRAHEDRON LETTERS 58 ( 10 ) 959 - 962 2017.03 [Refereed]
Enantioselective Mukaiyama-Michael Reaction of Cyclic alpha-Alkylidene beta-Keto Phosphine Oxide and Phosphonate and Asymmetric Synthesis of (R)-Homosarkomycin
Kotaro Nagatani, Atsushi Minami, Haruka Tezuka, Yunosuke Hoshino, Masahisa Nakada
ORGANIC LETTERS 19 ( 4 ) 810 - 813 2017.02 [Refereed]
SYNTHESIS OF A NEW CHIRAL C-2-SYMMETRIC NHC-AuCl COMPLEX
Naoya Okitsu, Takuya Yoshida, Kensuke Usui, Masahisa Nakada
HETEROCYCLES 92 ( 4 ) 720 - 732 2016.04 [Refereed]
Research on the design, synthesis, and catalytic activity of chiral N-heterocyclic carbene ligand-metal complexes
Kensuke Usui, Takuya Yoshida, Masahisa Nakada
TETRAHEDRON-ASYMMETRY 27 ( 2-3 ) 107 - 113 2016.02 [Refereed]
Highly enantioselective catalytic asymmetric Mukaiyama-Michael reactions of cyclic alpha-alkylidene beta-oxo imides
Harufumi Oyama, Kohei Orimoto, Takashi Niwa, Masahisa Nakada
TETRAHEDRON-ASYMMETRY 26 ( 5-6 ) 262 - 270 2015.03 [Refereed]
A highly stereoselective intramolecular Diels-Alder reaction for construction of the AB ring moiety of bruceantin
Kenji Usui, Takahiro Suzuki, Masahisa Nakada
TETRAHEDRON LETTERS 56 ( 10 ) 1247 - 1251 2015.03 [Refereed]
ENANTIOSELECTIVE TOTAL SYNTHESIS OF (+)-BUCIDARASINS A AND C
Kenji Usui, Masahisa Nakada
HETEROCYCLES 91 ( 2 ) 332 - 350 2015.02 [Refereed]
Highly enantioselective catalytic Friedel-Crafts reactions of cyclic alpha-alkylidene beta-oxo imides
Harufumi Oyama, Masahisa Nakada
TETRAHEDRON-ASYMMETRY 26 ( 4 ) 195 - 202 2015.02 [Refereed]
Enantioselective Approach to Polycyclic Polyprenylated Acylphloroglucinols via Catalytic Asymmetric Intramolecular Cyclopropanation
Yuta Uetake, Masahiro Uwamori, Masahisa Nakada
JOURNAL OF ORGANIC CHEMISTRY 80 ( 3 ) 1735 - 1745 2015.02 [Refereed]
Synthesis and characterization of a new C-2-symmetrical chiral tridentate N-heterocyclic carbene ligand coordinated Cr(III) complex
Yuta Uetake, Takashi Niwa, Masahisa Nakada
TETRAHEDRON-ASYMMETRY 26 ( 2-3 ) 158 - 162 2015.02 [Refereed]
Highly Enantioselective Catalytic Asymmetric [2+2] Cycloadditions of Cyclic alpha-Alkylidene beta-Oxo Imides with Ynamides
Kazuaki Enomoto, Harufumi Oyama, Masahisa Nakada
CHEMISTRY-A EUROPEAN JOURNAL 21 ( 7 ) 2798 - 2802 2015.02 [Refereed]
A CONCISE APPROACH TO TETRACYCLIC SPIROAMINE SCAFFOLD OF ERYTHRINAN ALKALOIDS VIA AN OXIDATIVE DEAROMATIZATION-SPIROCYCLIZATION SEQUENCE
Emi Saito, Akihiko Nakamura, Masahisa Nakada
HETEROCYCLES 90 ( 2 ) 1387 - 1395 2015.01 [Refereed]
Formal Total Synthesis of (-)-Taxol through Pd-Catalyzed Eight-Membered Carbocyclic Ring Formation
Sho Hirai, Masayuki Utsugi, Mitsuhiro Iwamoto, Masahisa Nakada
CHEMISTRY-A EUROPEAN JOURNAL 21 ( 1 ) 355 - 359 2015.01 [Refereed]
Synthesis of cycloalkanone-fused cyclopropanes by Au(I)-catalyzed oxidative ene-yne cyclizations
Yuta Uetake, Takashi Niwa, Masahisa Nakada
TETRAHEDRON LETTERS 55 ( 50 ) 6847 - 6850 2014.12 [Refereed]
Total Synthesis of (-)-Bucidarasin A Starting from an Original Chiral Building Block
Kenji Usui, Misaki Kanbe, Masahisa Nakada
ORGANIC LETTERS 16 ( 18 ) 4734 - 4737 2014.09 [Refereed]
Enantioselective total synthesis of (-)-cyathin B-2
Yu Kobayakawa, Masahisa Nakada
JOURNAL OF ANTIBIOTICS 67 ( 6 ) 483 - 485 2014.06 [Refereed]
Enantioselective total synthesis of (-)-cyathin B-2
Yu Kobayakawa, Masahisa Nakada
JOURNAL OF ANTIBIOTICS 67 ( 6 ) 483 - 485 2014.06 [Refereed]
Preparation of chiral building blocks for the enantioselective total synthesis of ent-kauranoids by the pig liver esterase-catalyzed asymmetric hydrolysis of a dialkyl malonate-type prochiral diester
Yuji Namiki, Tomohiro Fujii, Masahisa Nakada
TETRAHEDRON-ASYMMETRY 25 ( 9 ) 718 - 724 2014.05 [Refereed]
ENANTIOSELECTIVE TOTAL SYNTHESIS OF (-)-SCABRONINE D
Yu Kobayakawa, Masahisa Nakada
HETEROCYCLES 89 ( 3 ) 669 - 677 2014.03 [Refereed]
Direct reductive amination using triethylsilane and catalytic bismuth(III) chloride
Takehiko Matsumura, Masahisa Nakada
TETRAHEDRON LETTERS 55 ( 10 ) 1829 - 1834 2014.03 [Refereed]
Stereoselective construction of the ABC-ring system of fusidane triterpenes via intermolecular/transannular Michael reaction cascade
Tomohiro Fujii, Masahisa Nakada
TETRAHEDRON LETTERS 55 ( 9 ) 1597 - 1601 2014.02 [Refereed]
Preparation of imidazolinium salts by the Pd-catalyzed reduction of thioureas with triethylsilane and trialkylsilyl triflate
Takehiko Matsumura, Masahisa Nakada
TETRAHEDRON LETTERS 55 ( 8 ) 1412 - 1415 2014.02 [Refereed]
Enantioselective total syntheses of cyathane diterpenoids.
Nakada Masahisa
Enantioselective total syntheses of cyathane diterpenoids. 14 ( 4 ) 2014
Enantioselective Total Syntheses of Cyathane Diterpenoids
Nakada, Masahisa
CHEMICAL RECORD 14 ( 4 ) 641 - 662 2014
Highly stereoselective Michael reduction/intramolecular Michael reaction cascade to synthesize trans-stereodiad comprising an all-carbon quaternary stereogenic center
Tomohiro Fujii, Kohei Orimoto, Masahisa Nakada
TETRAHEDRON LETTERS 55 ( 5 ) 1100 - 1103 2014.01 [Refereed]
FACILE FORMATION OF IMIDAZOLINIUM SALT BY REACTION OF CORRESPONDING DIAMINE AND TRIMETHYL ORTHOFORMATE IN 1,1,1,3,3,3-HEXAFLUOROISOPROPANOL
Kensuke Usui, Masahisa Nakada
HETEROCYCLES 88 ( 2 ) 1539 - 1551 2014.01 [Refereed]
Total Syntheses of (-)-Scabronines G and A, and (-)-Episcabronine A
Yu Kobayakawa, Masahisa Nakada
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 52 ( 29 ) 7569 - 7573 2013.07 [Refereed]
Collective Total Synthesis of PPAPs: Total Synthesis of Clusianone via Intramolecular Cyclopropanation
Masahiro Uwamori, Masahisa Nakada
NATURAL PRODUCT COMMUNICATIONS 8 ( 7 ) 955 - 959 2013.07 [Refereed]
Stereoselective total synthesis of (±)-hyperforin via intramolecular cyclopropanation
Masahiro Uwamori, Masahisa Nakada
Tetrahedron Letters 54 ( 15 ) 2022 - 2025 2013.04
Research on the pig liver esterase (PLE)-catalyzed kinetic resolution of half-esters derived from prochiral diesters
Naoyoshi Noguchi, Kazuhiro Tsuna, Masahisa Nakada
TETRAHEDRON-ASYMMETRY 24 ( 7 ) 357 - 361 2013.04 [Refereed]
A short and enantioselective preparation of taxol A-ring fragment
Sho Hirai, Naoko Urushizako, Masayuki Miyano, Tomohiro Fujii, Masahisa Nakada
TETRAHEDRON LETTERS 54 ( 14 ) 1888 - 1892 2013.04 [Refereed]
PREPARATION OF IMIDES VIA THE PALLADIUM-CATALYZED COUPLING REACTION OF ORGANOSTANNANES WITH METHYL N-[METHOXY(METHYLTHIO)METHYLENE]CARBAMATE
Kohei Orimoto, Takuhei Tomizawa, Yuki Namera, Harufumi Oyama, Takashi Niwa, Masahisa Nakada
HETEROCYCLES 87 ( 4 ) 827 - + 2013.04 [Refereed]
Stereoselective total synthesis of garsubellin A
Masahiro Uwamori, Masahisa Nakada
JOURNAL OF ANTIBIOTICS 66 ( 3 ) 141 - 145 2013.03 [Refereed]
Enantioselective Total Synthesis of (+)-Colletoic Acid via Catalytic Asymmetric Intramolecular Cyclopropanation of an alpha-Diazo-beta-keto Diphenylphosphine Oxide
Takashi Sawada, Masahisa Nakada
ORGANIC LETTERS 15 ( 5 ) 1004 - 1007 2013.03 [Refereed]
Catalytic asymmetric [4 + 2] cycloadditions and Hosomi-Sakurai reactions of α-alkylidene β-keto imides
Kohei Orimoto, Harufumi Oyama, Yuki Namera, Takashi Niwa, Masahisa Nakada
Organic Letters 15 ( 4 ) 768 - 771 2013.02
Collective total synthesis of PPAPs: total synthesis of clusianone via intramolecular cyclopropanation.
Uwamori Masahiro, Nakada Masahisa
Collective total synthesis of PPAPs: total synthesis of clusianone via intramolecular cyclopropanation. 8 ( 7 ) 2013
Total syntheses of (-)-scabronines G and A, and (-)-episcabronine A.
Kobayakawa Yu, Nakada Masahisa
Total syntheses of (-)-scabronines G and A, and (-)-episcabronine A. 52 ( 29 ) 2013
Enantioselective total synthesis of (+)-ophiobolin A.
Tsuna Kazuhiro, Noguchi Naoyoshi, Nakada Masahisa
Enantioselective total synthesis of (+)-ophiobolin A. 19 ( 17 ) 2013
Enantioselective total synthesis of (+)-colletoic acid via catalytic asymmetric intramolecular cyclopropanation of an α-diazo-β-keto diphenylphosphine oxide.
Sawada Takashi, Nakada Masahisa
Enantioselective total synthesis of (+)-colletoic acid via catalytic asymmetric intramolecular cyclopropanation of an α-diazo-β-keto diphenylphosphine oxide. 15 ( 5 ) 2013
Stereoselective total synthesis of garsubellin A.
Uwamori Masahiro, Nakada Masahisa
Stereoselective total synthesis of garsubellin A. 66 ( 3 ) 2013
Catalytic asymmetric [4 + 2] cycloadditions and Hosomi-Sakurai reactions of α-alkylidene β-keto imides.
Orimoto Kohei, Oyama Harufumi, Namera Yuki, Niwa Takashi, Nakada Masahisa
Catalytic asymmetric [4 + 2] cycloadditions and Hosomi-Sakurai reactions of α-alkylidene β-keto imides. 15 ( 4 ) 2013
Allylic oxidations in natural product synthesis
Akihiko Nakamura, Masahisa Nakada
Synthesis (Germany) 45 ( 11 ) 1421 - 1451 2013
Preparation of Imides via the Palladium-Catalyzed Coupling Reaction of Organoborons with Methyl N-[Methoxy(methylthio)methylene]carbamate as a One-Carbon Elongation Reaction
Takuhei Tomizawa, Kohei Orimoto, Takashi Niwa, Masahisa Nakada
ORGANIC LETTERS 14 ( 24 ) 6294 - 6297 2012.12 [Refereed]
A Non-Heme Iron(III) Complex with Porphyrin-like Properties That Catalyzes Asymmetric Epoxidation
Takashi Niwa, Masahisa Nakada
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 134 ( 33 ) 13538 - 13541 2012.08 [Refereed]
Pd-catalyzed reductive cleavage of alkyl aryl sulfides with triethylsilane that is accelerated by trialkylsilyl chloride
Takehiko Matsumura, Takashi Niwa, Masahisa Nakada
TETRAHEDRON LETTERS 53 ( 33 ) 4313 - 4316 2012.08 [Refereed]
Stereoselective Total Synthesis of Nemorosone
Masahiro Uwamori, Aya Saito, Masahisa Nakada
JOURNAL OF ORGANIC CHEMISTRY 77 ( 11 ) 5098 - 5107 2012.06 [Refereed]
Asymmetric and Highly Stereoselective Synthesis of the DEF-Ring Moiety of (-)-FR182877 and Its Derivative Inducing Mitotic Arrest
Yu Kobayakawa, Yusuke Mori, Hideki Okajima, Yasuhiko Terada, Masahisa Nakada
ORGANIC LETTERS 14 ( 8 ) 2086 - 2089 2012.04 [Refereed]
Preparation of new chiral bisoxazoline ligands for the catalytic asymmetric intramolecular cyclopropanation of alpha-diazo-beta-keto phenyl sulfone to afford a useful bicyclo[3.1.0]hexane derivative
Takashi Sawada, Masahisa Nakada
TETRAHEDRON-ASYMMETRY 23 ( 5 ) 350 - 356 2012.03 [Refereed]
Synthetic studies on (+)-bucidarasin C: two diastereoselective transannular reactions producing cis-decaline derivatives that show reversal selectivity
Akinobu Nakahara, Misaki Kanbe, Masahisa Nakada
TETRAHEDRON LETTERS 53 ( 12 ) 1518 - 1522 2012.03 [Refereed]
Preparation of imides via the palladium-catalyzed coupling reaction of organoborons with methyl N-[methoxy(methylthio)methylene]carbamate as a one-carbon elongation reaction.
Tomizawa Takuhei, Orimoto Kohei, Niwa Takashi, Nakada Masahisa
Preparation of imides via the palladium-catalyzed coupling reaction of organoborons with methyl N-[methoxy(methylthio)methylene]carbamate as a one-carbon elongation reaction. 14 ( 24 ) 2012
A non-heme iron(III) complex with porphyrin-like properties that catalyzes asymmetric epoxidation.
Niwa Takashi, Nakada Masahisa
A non-heme iron(III) complex with porphyrin-like properties that catalyzes asymmetric epoxidation. 134 ( 33 ) 2012
Stereoselective total synthesis of nemorosone.
Uwamori Masahiro, Saito Aya, Nakada Masahisa
Stereoselective total synthesis of nemorosone. 77 ( 11 ) 2012
Asymmetric and highly stereoselective synthesis of the DEF-ring moiety of (-)-FR182877 and its derivative inducing mitotic arrest.
Kobayakawa Yu, Mori Yusuke, Okajima Hideki, Terada Yasuhiko, Nakada Masahisa
Asymmetric and highly stereoselective synthesis of the DEF-ring moiety of (-)-FR182877 and its derivative inducing mitotic arrest. 14 ( 8 ) 2012
Synthesis of medium-sized carbocyclic ketones via the intramolecular B-alkyl Liebeskind-Srogl coupling reaction
Kazuhiro Tsuna, Naoyoshi Noguchi, Masahisa Nakada
TETRAHEDRON LETTERS 52 ( 52 ) 7202 - 7205 2011.12 [Refereed]
Enantioselective Total Synthesis of (-)-FR182877
Natsumi Tanaka Suzuki, Takahiro Suzuki, Takehiko Matsumura, Yousuke Hosoya, Tomoyuki Nakazato, Masahisa Nakada
JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN 69 ( 6 ) 646 - 660 2011.06 [Refereed]
Enantioselective Total Synthesis of (-)-FR182877
TANAKA SUZUKI Natsumi, SUZUKI Takahiro, MATSUMURA Takehiko, HOSOYA Yousuke, NAKAZATO Tomoyuki, NAKADA Masahisa
J. Synth. Org. Chem. Jpn. 69 ( 6 ) 646 - 660 2011.06 [Refereed]
Convergent total synthesis of (+)-ophiobolin A.
Tsuna Kazuhiro, Noguchi Naoyoshi, Nakada Masahisa
Convergent total synthesis of (+)-ophiobolin A. 50 ( 40 ) 2011
Convergent Total Synthesis of (+)-Ophiobolin A
Kazuhiro Tsuna, Naoyoshi Noguchi, Masahisa Nakada
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 50 ( 40 ) 9452 - 9455 2011 [Refereed]
Enantioselective divergent approaches to both (-)-platensimycin and (-)-platencin
Sho Hirai, Masahisa Nakada
TETRAHEDRON 67 ( 2 ) 518 - 530 2011.01 [Refereed]
An enantioselective approach to (-)-platencin via catalytic asymmetric intramolecular cyclopropanation
Sho Hirai, Masahisa Nakada
TETRAHEDRON LETTERS 51 ( 38 ) 5076 - 5079 2010.09 [Refereed]
Synthetic studies on nemorosone via enantioselective intramolecular cyclopropanation
Masahito Abe, Aya Saito, Masahisa Nakada
TETRAHEDRON LETTERS 51 ( 9 ) 1298 - 1302 2010.03 [Refereed]
Synthesis of NH006--a photostable fungicide effective against Botrytis cinerea--according to the asymmetric total synthesis of MK8383.
Hayashi Nobuyuki, Yamamoto Kentaro, Minowa Nobuto, Mitomi Masaaki, Nakada Masahisa
Synthesis of NH006--a photostable fungicide effective against Botrytis cinerea--according to the asymmetric total synthesis of MK8383. 8 ( 8 ) 2010
Synthesis of NH006-a photostable fungicide effective against Botrytis cinerea-according to the asymmetric total synthesis of MK8383
Nobuyuki Hayashi, Kentaro Yamamoto, Nobuto Minowa, Masaaki Mitomi, Masahisa Nakada
ORGANIC & BIOMOLECULAR CHEMISTRY 8 ( 8 ) 1821 - 1825 2010 [Refereed]
Synthetic studies on the taxane skeleton: effective construction of eight-membered carbocyclic ring by palladium-catalyzed intramolecular alpha-alkenylation of a methyl ketone
Masayuki Utsugi, Yasuaki Kamada, Masahisa Nakada
TETRAHEDRON LETTERS 49 ( 32 ) 4754 - 4757 2008.08 [Refereed]
Synthetic Studies on (–)-Scabronine A
Watanabe, H, Nakada, M
Tetrahedron Lett. 49 1518 - 1522 2008 [Refereed]
Biomimetic Total Synthesis of (–)-Erinacine E
Watanabe, H, Nakada, M
J. Am. Chem. Soc. 130 1150 - 1151 2008 [Refereed]
Catalytic asymmetric Nozaki-Hiyama reactions with a tridentate Bis(oxazolinyl)carbazole ligand
Masahiro Inoue, Takahiro Suzuki, Akihiro Kinoshita, Masahisa Nakada
CHEMICAL RECORD 8 ( 3 ) 169 - 181 2008 [Refereed]
Synthetic studies on (-)-FR182877: construction of the ABCD ring system via the intramolecular cycloadditions (1)
Takahiro Suzuki, Natsumi Tanaka, Takehiko Matsumura, Yosuke Hosoya, Masahisa Nakada
TETRAHEDRON LETTERS 48 ( 37 ) 6483 - 6487 2007.09 [Refereed]
Synthetic studies on (-)-FR182877: construction of the ABCD ring system via the intramolecular cycloadditions (2)
Natsumi Tanaka, Takahiro Suzuki, Yosuke Hosoya, Masahisa Nakada
TETRAHEDRON LETTERS 48 ( 37 ) 6488 - 6492 2007.09 [Refereed]
Construction of the taxane skeleton via the stereoselective conjugate addition of cyanide and the intramolecular B-alkyl Suzuki-Miyaura coupling reaction
Masayuki Utsugi, Yasuaki Kamada, Hidetoshi Miyamoto, Masahisa Nakada
TETRAHEDRON LETTERS 48 ( 39 ) 6868 - 6872 2007.09 [Refereed]
Highly enantioselective preparation of tricyclo[4.4.0.0(5,7)]decene derivatives via catalytic asymmetric intramolecular cyclopropanation reactions of alpha-diazo-beta-keto esters
Ryoji Ida, Masahisa Nakada
TETRAHEDRON LETTERS 48 ( 28 ) 4855 - 4859 2007.07 [Refereed]
Synthetic studies on phloroglucins: a new approach to the bicyclo[3.3.1]nonane system via the regioselective ring-opening of the methoxycyclopropane
Masahito Abe, Masahisa Nakada
TETRAHEDRON LETTERS 48 ( 28 ) 4873 - 4877 2007.07 [Refereed]
New preparation of tridentate bis-oxazoline carbazole ligand effective for enantioselective Nozaki-Hiyama reaction
Masahiro Inoue, Masahisa Nakada
HETEROCYCLES 72 133 - 138 2007.04 [Refereed]
Catalytic asymmetric intramolecular cyclopropanation of 2-diazo-3-oxo-6-heptenoic acid esters
Hiroyuki Takeda, Masahiro Honma, Ryoji Ida, Takashi Sawada, Masahisa Nakada
SYNLETT ( 4 ) 579 - 582 2007.03 [Refereed]
抗腫瘍性化合物Taxolの不斉全合成研究:エポキシドに対しての1,5-ヒドリドシフトによるtrans縮環したB,C環部位構築
日本薬学会第127年会 2007.03
(+)-ophiobolin Aの不斉全合成研究
日本薬学会第127年会 2007.03
エリナシンBの不斉全合成
日本薬学会第127年会 2007.03
(-)-タキソールの不斉全合成研究
日本化学会第87春季年会 2007.03
(-)-FR182877の全合成研究
日本化学会第87春季年会 2007.03
(-)-physostigmineの形式全合成
日本化学会第87春季年会 2007.03
ハイパーフォリンの不斉全合成研究
日本化学会第87春季年会 2007.03
Enantioselective Total Synthesis of (–)-Erinacine B
Watanabe, H, Takano, M, Umino, A, Ito, T, Ishikawa, H, Nakada, M
Org. Lett. 9 359 - 362 2007 [Refereed]
Convergent Total Synthesis of (+)-Digitoxigenin via Catalytic Asymmetric Intramolecular Cyclopropanation
Honma, M, Nakada, M
Tetrahedron Lett. 48 1541 - 1544 2007
Structure Elucidation and Enantioselective, Protecting Group-Free Total Synthesis of the HMG-CoA Reductase Inhibitor, FR901512 via Catalytic Asymmetric Nozaki−Hiyama Reactions
Inoue, M, Nakada, M
J. Am. Chem. Soc 129 4164 - 4165 2007 [Refereed]
(+)-Digitoxigeninの全合成
第32回反応と合成の進歩シンポジウム 2006.12
光学活性多環式天然物の全合成研究
特定領域研究第三回公開シンポジウム 2006.12
ASYMMETRIC TOTAL SYNTHESIS OF BIOACTIVE POLYCYCLIC NATURAL PRODUCTS
9th International Symposium for Chinese Organic Chemists 2006.12
Studies on the structure-enantioselectivity relationships in the catalytic asymmetric intramolecular cyclopropanation reaction of alpha-diazo-beta-keto sulfones possessing a methyl-substituted phenyl group
Hiroyuki Takeda, Masahisa Nakada
TETRAHEDRON-ASYMMETRY 17 ( 20 ) 2896 - 2906 2006.11 [Refereed]
Hyperforinの不斉全合成研究
第90回有機合成シンポジウム 2006.11
触媒的不斉野崎ー檜山反応の開発とHMG-CoA還元酵素阻害剤FR901512の不斉全合成
第48回天然有機化合物討論会 2006.10
New construction of the bicyclo[3.3.1]nonane system via Lewis acid promoted regioselective ring-opening reaction of the tricyclo[4.4.0.0(5,7)]dec-2-ene derivative
Masahito Abe, Masahisa Nakada
TETRAHEDRON LETTERS 47 ( 36 ) 6347 - 6351 2006.09 [Refereed]
Asymmetric total synthesis of enantiopure (-)-methyl jasmonate via catalytic asymmetric intramolecular cyclopropanation of alpha-diazo-beta-keto sulfone
Hiroyuki Takeda, Hideaki Watanabe, Masahisa Nakada
TETRAHEDRON 62 ( 34 ) 8054 - 8063 2006.08 [Refereed]
Synthetic studies on taxol: Highly stereoselective construction of the taxol C-ring via S(N)2 ' reduction of an allylic phosphonium salt
Masayuki Utsugi, Masayuki Miyano, Masahisa Nakada
ORGANIC LETTERS 8 ( 14 ) 2973 - 2976 2006.07 [Refereed]
STUDIES ON ASYMMETRIC TOTAL SYNTHESIS OF (-)-FR182877
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
STUDIES ON ASYMMETRIC TOTAL SYNTHESIS OF HYPERFORIN
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
STEREOCONTROLLED TOTAL SYNTHESIS OF (+)-FR901516
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
STUDIES ON ASYMMETRIC TOTAL SYNTHESIS OF TAXOL
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
SYNTHETIC STUDIES ON (-)-SCABRONINE A
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
TOTAL SYNTHESIS OF NATURAL PRODUCTS VIA CATALYTIC ASYMMETRIC INTRAMOLECULAR CYCLOPROPANATION
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
SYNTHETIC STUDIES ON ENANTIOPURE (+)-DIGITOXIGENIN
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
STUDIES ON ENANTIOSELECTIVE TOTAL SYNTHESIS OF (+)-OPHIOBOLIN A
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
FURTHER SYNTHETIC STUDIES ON (+)-PHOMOPSIDIN
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
SYNTHETIC STUDIES ON ERINACINES
International Conference on Biodiversity and Natural Products (ICOB-5 & ISCNP-25 IUPAC) 2006.07
Synthetic studies on (+)-ophiobolin A: Asymmetric synthesis of the spirocyclic CD-ring moiety
N Noguchi, M Nakada
ORGANIC LETTERS 8 ( 10 ) 2039 - 2042 2006.05 [Refereed]
Synthetic Studies on Erinacines
The International Symposium on Chemistry, Biology & Medicine in Paphos, Cyprus 2006.05
Studies on the diastereoselectivity in the IMDA reactions of terminally activated (E,E,E)-nona-1,6,8-trienes
T Suzuki, N Tanaka, T Matsumura, Y Hosoya, M Nakada
TETRAHEDRON LETTERS 47 ( 10 ) 1593 - 1598 2006.03 [Refereed]
新規キラルビルディングブロックスの創製と
日本化学会第86春季年会 2006.03
(+)-ブシダラシンCの全合成研究
日本化学会第86春季年会 2006.03
(+)-ジギトキシゲニンの合成研究
日本化学会第86春季年会 2006.03
FR182877の全合成研究
日本化学会第86春季年会 2006.03
(-)-ブルセアンチンの全合成研究
日本化学会第86春季年会 2006.03
(-)-サイアンチウィジンFの全合成研究
日本化学会第86春季年会 2006.03
Hyperforinの全合成研究
日本化学会第86春季年会 2006.03
hirsuteneの全合成研究
日本化学会第86春季年会 2006.03
(+)-ホモプシジンの不斉全合成研究
日本化学会第86春季年会 2006.03
(+)-オフィオボリンAの不斉全合成研究
日本化学会第86春季年会 2006.03
FR901512の立体選択的合成研究
日本化学会第86春季年会 2006.03
(-)‐マリンゴライドの不斉全合成
日本化学会第86春季年会 2006.03
(+)-グアナカステペンAの不斉全合成研究
日本化学会第86春季年会 2006.03
Studies into asymmetric catalysis of the Nozaki-Hiyama allenylation
M Inoue, M Nakada
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 45 ( 2 ) 252 - 255 2006 [Refereed]
Studies on enantioselective total synthesis of Taxol
PACIFICHEM2005 2005.12
Synthetic studies on erinacines
PACIFICHEM2005 2005.12
Asymmetric catalysis on the intramolecular cyclopropanation of α-diazo-β-keto sulfones and synthetic studies on (+)-digitoxigenin
PACIFICHEM2005 2005.12
Catalytic asymmetric Nozaki-Hiyama reactions with a new chiral carbazole lligand
PACIFICHEM2005 2005.12
(-)-scabronine Aの収束的不斉全合成研究
PACIFICHEM2005 2005.12
Total Synthesis of (-)-Malyngolide via Catalytic Asymmetric Intramolecular Cyclopropanation
Heterocycles 66 2005.12
生物活性多環式天然物の不斉全合成
平成17年度秋季有機合成化学講習会 2005.11
生物活性多環式天然物の全合成研究
特定領域研究第一回公開シンポジウム 2005.11
タキソールの不斉全合成研究
第31回反応と合成の進歩シンポジウム 2005.11
Asymmetric Catalysis of Intramolecular Cyclopropanation of 5-Aryl-1-arylsulfonyl-1-diazo-5-hexene-2-ones
Adv. Synth. Catal. 347 1527 - 1532 2005.11
新規光学活性カルバゾール配位子を用いた触媒的不斉野崎檜山反応
第52回有機金属化学討論会 2005.10
Erinacine類の不斉全合成研究
第47回天然有機化合物討論会 2005.10
生物活性多環式天然物の全合成研究
第36回中部化学関係学協会支部連合秋季大会特別討論会:有機化学の新潮流 2005.09
生物活性多環式天然物の効率的不斉全合成研究
第10回PharmaScienceフォーラム 2005.09
Preparation of new chiral building blocks: Highly enantioselective reduction of prochiral 1,3-cycloalkanediones possessing a methyl group and a protected hydroxymethyl group at their C2 position with baker's yeast or CBS catalyst
H Watanabe, M Iwamoto, M Nakada
JOURNAL OF ORGANIC CHEMISTRY 70 ( 12 ) 4652 - 4658 2005.06 [Refereed]
サイアタンジテルペノイド類の不斉全合成研究
第87回有機合成シンポジウム 2005.06
生物活性多環式天然物の合成研究
第1回バイオメディカルフォーラム 2004.12
Development of silicon-tethered anionic reaction and its application to the synthesis of chiral A-ring moieties of Taxol (TM)
M Iwamoto, M Miyano, M Utsugi, H Kawada, M Nakada
TETRAHEDRON LETTERS 45 ( 47 ) 8647 - 8651 2004.11 [Refereed]
Synthetic studies on the seven- and eight-membered rings by the intramolecular Nozaki-Hiyama reaction of the allylic phosphates
M Iwamoto, M Miyano, M Utsugi, H Kawada, M Nakada
TETRAHEDRON LETTERS 45 ( 47 ) 8653 - 8657 2004.11 [Refereed]
Synthetic studies on the taxane skeleton: Construction of eight-membered carbocyclic rings by the intramolecular B-alkyl Suzuki-Miyaura cross-coupling reaction
H Kawada, M Iwamoto, M Utsugi, M Miyano, M Nakada
ORGANIC LETTERS 6 ( 24 ) 4491 - 4494 2004.11 [Refereed]
Development of silicon-tethered anionic reaction and its application to the synthesis of chiral A-ring moieties of Taxol (TM)
M Iwamoto, M Miyano, M Utsugi, H Kawada, M Nakada
TETRAHEDRON LETTERS 45 ( 47 ) 8647 - 8651 2004.11 [Refereed]
Synthetic studies on the seven- and eight-membered rings by the intramolecular Nozaki-Hiyama reaction of the allylic phosphates
M Iwamoto, M Miyano, M Utsugi, H Kawada, M Nakada
TETRAHEDRON LETTERS 45 ( 47 ) 8653 - 8657 2004.11
Synthetic studies on the taxane skeleton: Construction of eight-membered carbocyclic rings by the intramolecular B-alkyl Suzuki-Miyaura cross-coupling reaction
H Kawada, M Iwamoto, M Utsugi, M Miyano, M Nakada
ORGANIC LETTERS 6 ( 24 ) 4491 - 4494 2004.11 [Refereed]
不斉リガンド創出に基づく不斉触媒反応の開発と天然物合成への応用
有機合成化学ミニシンポジウム,東京工業大学,大岡山,東京 2004.09
Studies on catalytic asymmetric Nozaki-Hiyama propargylation
M Inoue, M Nakada
ORGANIC LETTERS 6 ( 17 ) 2977 - 2980 2004.08 [Refereed]
Studies on catalytic asymmetric Nozaki-Hiyama propargylation
M Inoue, M Nakada
ORGANIC LETTERS 6 ( 17 ) 2977 - 2980 2004.08
新規光学活性三座配位子を用いた触媒的不斉野崎—檜山プロパルギル化反応
日本化学会第84春季年会 神戸 2004.03
サイアチン類の合成研究(1)
日本化学会第84春季年会 神戸 2004.03
サイアチン類の合成研究(2)
日本化学会第84春季年会 神戸 2004.03
触媒的不斉分子内シクロプロパン化反応の研究(1)
日本化学会第84春季年会 神戸 2004.03
触媒的不斉分子内シクロプロパン化反応の研究(2)
日本化学会第84春季年会 神戸 2004.03
タキサン骨格の合成法研究(1)
日本化学会第84春季年会 神戸 2004.03
タキサン骨格の合成法研究(2)
日本化学会第84春季年会 神戸 2004.03
不斉触媒を用いた新規キラルシントンの合成
日本化学会第84春季年会 神戸 2004.03
(-)-FR182877の全合成研究
日本化学会第84春季年会 神戸 2004.03
(+)-ホモプシジンの全合成
日本化学会第84春季年会 神戸 2004.03
First total synthesis of antimitotic compound, (+)-phomopsidin
T Suzuki, K Usui, Y Miyake, M Namikoshi, M Nakada
ORGANIC LETTERS 6 ( 4 ) 553 - 556 2004.02 [Refereed]
First total synthesis of antimitotic compound, (+)-phomopsidin
T Suzuki, K Usui, Y Miyake, M Namikoshi, M Nakada
ORGANIC LETTERS 6 ( 4 ) 553 - 556 2004.02 [Refereed]
Synthetic Studies on Erinacines: Enantioselective Total Synthesis of (+)-Allocycthin B2
Org. Lett. 6 4897 - 4900 2004
Synthetic Studies on Erinacines: Enantioselective Total Synthesis of (+)-Allocycthin B2
Org. Lett. 6 4897 - 4900 2004 [Refereed]
α-ジアゾ-β-ケトスルホン類の触媒的不斉分子内シクロプロパン化反応の研究
第84回有機合成シンポジウム 2003.11
新規光学活性三座配位子を用いた触媒的不斉野崎ー檜山アリル化反応
第29回反応と合成の進歩シンポジウム 2003.10
抗腫瘍性抗生物質phomopsidineの全合成研究
第45回天然有機化合物討論会 2003.10
タキサン骨格の合成法研究(2)
日本化学会第83春季年会、東京 2003.03
New asymmetric tridentate carbazole ligand: Its preparation and application to Nozaki-Hiyama allylation
T Suzuki, A Kinoshita, H Kawada, M Nakada
SYNLETT ( 4 ) 570 - 572 2003.03 [Refereed]
サイアチン骨格の合成研究
日本化学会第83春季年会、東京 2003.03
触媒的不斉分子内シクロプロパン化反応の研究(1)
日本化学会第83春季年会、東京 2003.03
触媒的不斉分子内シクロプロパン化反応の研究(2)
日本化学会第83春季年会、東京 2003.03
触媒的不斉分子内シクロプロパン化反応の研究(3)
日本化学会第83春季年会、東京 2003.03
タキサン骨格の合成法研究(1)
日本化学会第83春季年会、東京 2003.03
タキサン骨格の合成法研究(2)
日本化学会第83春季年会、東京 2003.03
新規光学活性三座配位子を用いた触媒的不斉野崎-檜山アリル化反応(1)
日本化学会第83春季年会、東京 2003.03
新規光学活性三座配位子を用いた触媒的不斉野崎-檜山アリル化反応(2)
日本化学会第83春季年会、東京 2003.03
Asymmetric catalysis of Nozaki-Hiyama allylation and methallylation with a new tridentate bis(oxazolinyl)carbazole ligand
M Inoue, T Suzuki, M Nakada
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY 125 ( 5 ) 1140 - 1141 2003.02 [Refereed]
A New Preparation of Cyclic Sulfates: A Highly 1,3-Asymmetric Induction in Halocyclosulfations
Synth. Commun. 33 2857 - 2866 2003
Asymmetric Catalysis on the Intramolecular Cyclopropanations of α-Diazo-β-keto Sulfones
J. Am. Chem. Soc. 125 2860 - 2861 2003 [Refereed]
Preparation of New Chiral Building Blocks via Asymmetric Catalysis
Tetrahedron Lett. 44 7239 - 7244 2003 [Refereed]
Enantioselective Intramolecular Cyclopropanation of α-Diazo-β-keto Sulfones: Asymmetric Synthesis of
Tetrahedron Lett. 44 9007 - 9011 2003 [Refereed]
Asymmetric Catalysis of Nozaki-Hiyama Allylation and Methallylation with A New Tridentate Bis(oxazolinyl)carbazole Ligand
J. Am. Chem. Soc. 125 2003 [Refereed]
A New Asymmetric Tridentate Carbazole Ligand: Its Preparation and Application to Nozaki-Hiyama Allylation
SYNLETT 2003
Synthetic Studies on the Cyathin Core
The 9th International Conference on New Aspects of Organic Chemistry (IKCOC-9) (Kyoto Park Hotel, Kyoto, Japan, November 10-14, 2003), Prof. Emeritus, Zen-ichi Yoshida, ed. The Kinki Chemical Society, Japan 2003
Synthetic Studies on Taxane Skeleton
The 9th International Conference on New Aspects of Organic Chemistry (IKCOC-9) (Kyoto Park Hotel, Kyoto, Japan, November 10-14, 2003), Prof. Emeritus, Zen-ichi Yoshida, ed. The Kinki Chemical Society, Japan 2003
A New Preparation of Cyclic Sulfates: A Highly 1,3-Asymmetric Induction in Halocyclosulfations
Synth. Commun. 33 2003
Asymmetric Catalysis on the Intramolecular Cyclopropanations of α-Diazo-β-keto Sulfones
J. Am. Chem. Soc. 125 2003 [Refereed]
Preparation of New Chiral Building Blocks via Asymmetric Catalysis
Tetrahedron Lett. 44 2003 [Refereed]
Enantioselective Intramolecular Cyclopropanation of α-Diazo-β-keto Sulfones: Asymmetric Synthesis of Bicyclo[4.1.0]heptanes and Tricyclo[4.4.0.0]decenes
Tetrahedron Lett. 44 2003 [Refereed]
配位子及び不斉触媒
特願出 2002-367304号 2002.12
新規ハロ環状硫酸エステル化反応とそのジアステレオ選択性の研究
日本化学会第81春季年会, 東京 2002.03
FR182877の全合成研究(1)
日本化学会第81春季年会, 東京 2002.03
FR182877の全合成研究(1)
日本化学会第81春季年会, 東京 2002.03
FR182877の全合成研究(2)
日本化学会第81春季年会, 東京 2002.03
Sgnthetic Studies on FR182877 : An Asymmetric Synthesis of the AB Ring Moiety of FR182877 via a Dias teieo selective Intramolecular Diels-Alder Reaction
Tetrahedron Letl. 43 3263 - 3267 2002
Synthetic Studies on FR182877
8th International Conference on Chemistry of Antibiotics and Related Microbial Products (Tokyo, Japan, October 21-25 2002), S. Ōmura and K. Tatsuta, ed., National Organizing Committee of ICCA-8 2002
Synthetic Studies on an Antitumor Cyclic Peptide, Ustiloxin A
18th International Congress of Heterocyclic Chemistry (Pacifico Yokohama, Japan, July29-August 3, 2001), M. Shibasaki, ed., International Society of Heterocyclic Chemistry 2002
Synthetic Studies on FR182877: An Asymmetric Synthesis of the AB Ring Moiety of FR182877 via a Diastereoselective Intramolecular Diels-Alder Reaction
Tetrahedron Letters 43 2002 [Refereed]
Synthetic Studies on an Antitumor Cyclic Peptide, Ustiloxin A.
18th International Congress of Heterocyclic Chemistry, Pacifico Yokohama, Japan. 2001.07
フォモプシジンの合成研究
日本化学会第79春季年会2001年講演予稿集/日本化学会 2001.03
タキサン骨格の合成研究
日本化学会第79春季年会2001年講演予稿集/日本化学会 2001.03
ウスチロキシンAの合成研究
日本化学会第79春季年会2001年講演予稿集/日本化学会 2001.03
不斉分子内シクロプロパン化反応の研究
日本化学会第79春季年会2001年講演予稿集/日本化学会 2001.03
C,O-アセト酢酸エステルジアニオンによるTHF,THP誘導体のワンポット合成
日本化学会第79春季年会2001年講演予稿集/日本化学会 2001.03
FR182877の全合成研究
日本化学会第79春季年会2001年講演予稿集/日本化学会 2001.03
光学活性テトラヒドロフラン、ピラン誘導体の新規合成法研究
日本化学会第78春季年会2000年講演予稿集/日本化学会 2000.03
新規ルートによるタキサン骨格の合成法研究
日本化学会第78春季年会2000年講演予稿集/日本化学会 2000.03
Preparation of Novel Synthons, Uniquely Functionalized Tetrahydrofuran and Tetrahydropyran Derivatives
Chem. Pharm. Bull. 48/,1581 2000
Effect of Amines of the Selective Bromination of Some β-Substituted-2-butenoic Esters
Synth. Commun. 30 863 - 868 2000 [Refereed]
Effect of Amines of the Selective Bromination of Some β-Substituted-2-butenoic Esters.
Synth. Commun. 30 2000 [Refereed]
Preparation of Novel Synthons, Uniquely Functionalized Tetrahydrofuran and Tetrahydropyran Derivatives
Chem. Pharm. Bull. 48/,1581 2000 [Refereed]
タキサン骨格の合成研究
日本化学会第76春季年会1999年講演予稿集II/日本化学会 1999.03
光学活性テトラヒドロフラン、ピラン誘導体の新規合成法研究
日本化学会第76春季年会1999年講演予稿集II/日本化学会 1999.03
Reaction of dianions of acetoacetic esters with epibromohydrin derivatives : A novel synthesis of tetrahydrofuran derivatives and tetrahydropyran
Tetrahedron Letters' 40/,9077-9080 1999 [Refereed]
Reaction of dianions of acetoacetic esters with epibromohydrin derivatives : A novel synthesis of tetrahydrofuran derivatives and tetrahydropyran derivatives
Tetrahedron Lett./Elsevier Science 40 1999 [Refereed]
タキソールの不斉全合成研究—C環部位の立体選択的合成—
日本化学会第74春季年会/日本化学会 1998.03
光学活性シクロヘキサノン類のワンポット合成
日本化学会第74春季年会/日本化学会 1998.03
A Concise Synthetic Approach to Taxol C-Ring Fragment
Tetrahedron Lett. 39/,313 1998 [Refereed]
A Concise Synthetic Approach to Taxol C-Ring Fragment
Tetrahedron Lett./Elsevier Science Ltd 39;3/4 PP313-316 1998 [Refereed]
A Concise Synthetic Approach to Taxol C-Ring Fragment
Tetrahedron Lett./Elsevier Science Ltd 39;3/4(313) 1998.01 [Refereed]
タキソール類の合成—C環部位の効率的合成法の開発—
第33回有機合成化学協会関東支部(神奈川)シンポジウム/有機合成化学協会 1997.05
Synthesis, Structure-Activity Relationships, and Bioorganic Research of Homologs of Antitumor Macrolide, Rhizoxin Based on the Total Synthesis, and Development of Catalytic Asymmetric Synthesis for the Further Studies
Advances in Pharmaceutical Sciences 13/37-47 1997
Total Synthesis of Antitumor Macrolide, Rhizoxin and Chemistry of Acylsilane
Yakugaku Zasshi-J. Pharm. Soc. Jpn. 117 ( 486 ) 508 1997
Total Synthesis of Antitumor Macrolide, Rhizoxin and Chemistry of Aeylsilane
J.Pharm.Soc.Jpn. 117;486-508 ( 486 ) 508 1997
The First Chemical Synthesis of Wortmannin by Starting from Hydrocortisone
Tetrahedron Lett. 37/,6141 1996 [Refereed]
Total Synthesis of (+)-Tautomycin
Tethrahedron 52/,13363 1996 [Refereed]
The First Chemical Synthesis of Wortmannin by Starting from Hydrocortisone
Tetrahedron Lett./Elsevier Science Ltd 37 1996 [Refereed]
抗腫瘍性マクロリド、リゾキシンの構造活性相関研究(1)
日本化学会第72春季年会1997年講演予稿集II/日本化学会 1996
タキソール類の合成(1)ーC環部位の効率的合成法の開発ー
日本化学会第72春季年会1997年講演予稿集II/日本化学会 1996
トウトマイシンおよびトウトマイセチンの全合成研究
第70回有機合成シンポジウム講演要旨集/有機合成化学協会 1996
PI3-Kinase阻害剤Wortmanninの初の化学合成とbiological tool への展開
第69回有機合成シンポジウム講演要旨集/有機合成化学協会 1996
抗腫瘍性マクロリド、リゾキシンの全合成とアシルシランの化学
日本薬学会第117年会講演要旨集1/日本薬学会 1996
Total Synthesis of (+)-Tautomycin
Tetrahedron/Elsevier Science Ltd 52 1996 [Refereed]
Radiolabeling of Catalytic Subunits of PI3-Kinases with 17β-Hydroxy-16α-(125I)iodowortmannin: Identification of Gβγ-sensitive isoform as a complex composed of 46-kDa and 100-kDa subunits
Biochem. Biophys. Res. Commun./Academic Press 216;2 1995.02
抗腫瘍性マクロリド,リゾキシンの全合成
有機合成化学協会誌/有機合成化学協会 53 122 - 137 1995.02
Radiolabeling of Catalytic Subumits of PI3-Kinases with 17B-Hydroxy-16a-[125I]iodowortmanin : Identification of GBr-sensitive isoform as a complex compound of 46-KDa and 110-KDa subunits
Biochem. Biophys. Res. Commun. /216,655-661 1995
Radiolabeling of Catalytic Subumits of PI3-Kinases with 17B-Hydroxy-16a-[125I]iodowortmanin : Identification of GBr-sensitive isoform as a complex compound of 46-KDa and 110-KDa subunits
Biochem. Biophys. Res. Commun. /216,655-661 1995
Total Synthesis of Toxal. 2. Construction of A and C Ring Intermediates and Initial Attempts To Construct the ABC Ring System
J. Am. Chem. Soc. 117/,634-644 1995 [Refereed]
The First Total Synthesis of Antitumor Macrolide, Rhizoxin
Memories of the School of Science & Engineering /59,167-195 1995 [Refereed]
Radiolabeling of Catalytic Subumits of PI3-Kinases with 17B-Hydroxy-16a-[125I]iodowortmanin : Identification of GBr-sensitive isoform as a complex compound of 46-KDa and 110-KDa subunits
Biochem. Biophys. Res. Commun. /216,655-661 1995 [Refereed]
17B-Hydroxy-16a-[125I] indowortmanin, A Sensitive Labelling Agent for PI3-Kinases
Chem. Pham. Bull. /43,2276-2278 1995 [Refereed]
キラルなジアミンリガンド1を用いた触媒的不斉Diels-Alder反応
日本薬学会第116年会講演要旨集/日本薬学会第116年会実行委員会 1995
ホスファターゼ阻害物質トウトマイシンの全合成
日本薬学会第116年会講演要旨集/日本薬学会第116年会実行委員会 1995
Wortmannin の合成研究(2)
日本薬学会第116年会講演要旨集/日本薬学会第116年会実行委員会 1995
PI3-kinase阻害剤Wortmannin及びPI3-kinaseのBiological toolの合成研究
第37回天然有機化合物討論会講演要旨集/第37回天然有機化合物討論会実行委員会 1995
17β-Hydroxy-16α-(125I)iodowortmannin, A Sensitive Labelling Agent for PI3-Kinases
Chem. Pharm. Bull./Pharmaceutical Society of Japan 43;12 1995 [Refereed]
Total Synthesis of Taxol. 2. Construction of A and C Ring Intermediates and Initial Attempts To Construct the ABC Ring System
J. Am. Chem. Soc./American Chemical Society 117 1995 [Refereed]
The Total Synthesis of Antitumor Macrolide, Rhizoxin
Memoirs of the School of Science & Engineering/Waseda University 59 1995 [Refereed]
Non-chelation Controlled 1,3-Asymmetric Induction in β-Chiral Acylsilanes
Tetrahedron Lett. 35/,741-744 1994 [Refereed]
Calicheamicin θI1 : A Rationally Designed Molecule with Extremely Potent and Selective DNA Cleaving Properties and Apoptosis Inducing Activity
Angew. Chem. Int. Ed. Engl. 33/,183-186 1994 [Refereed]
The First Total Synthesis of the Antitumor Macrolide Rhizoxin:Synthesis of the Key Building Blocks
Tetrahedron Lett. 34/,1035-1038 1993 [Refereed]
Synthetic Study on an Antitumor Antibiotic Rhizoxin Using an Enzymatic Process on Prochiral β-Substituted Glutarates
Indian J. Chem. 32B/,159-162 1993 [Refereed]
The First Total Synthesis of the Antitumor Macrolide, Rhizoxin
Tetrahedron Lett. 34/,1039-1042 1993 [Refereed]
Total Synthesis of Calicheamicin γ1I. 3. The Final Stages
J. Am. Chem. Soc. 115/,7625-7635 1993 [Refereed]
Synthesis of ABC Taxoid Ring Systems via a Convergent Strategy
J. Chem. Soc. Chem. Commun. 12/,1024-1026 1993 [Refereed]
Synthetic Study on an Antitumor Antibiotic Rhizoxin Using an Enzymatic Process on Prochiral β-Substituted Glutarates
Pure Appl. Chem. 64/,1121-1124 1992 [Refereed]
Total Synthesis of Calicheamicin γ1I
J. Am. Chem. Soc. 114/,10082-10084 1992 [Refereed]
A Novel Synthesis of Acylsilanes
Tetrahedron Lett. 32/,4929-4932 1991 [Refereed]
Enantioselective Hydrolysis of Dialkyl 3-Monosubstituted Glutarates with Pig Liver Esterase
Structure-Optical Purity Relationships, Tetrahedron Lett. 29/,3951-3954 1988
High Diastereofacial Selectivity in Nucleophilic Additions to Chiral Acylsilanes
J. Am. Chem. Soc. 110/,4826-4827 1988 [Refereed]
PSJ(Phamaceutical Society of Japan) Award for Young Scientists
First Total Synthesis of Antimitotic Compound, (+)-Phomopsidin
Fifteenth International Conference on Organic Synthesis (ICOS-15) (August 1-6, 2004, Nagoya, Japan), Prof. Minoru Isobe and Hisashi Yamamoto, ed. Organizng Committee of ICOS-15, International Union of Pure and Applied Chemistry (IUPAC)
Synthetic Studies on Taxol
Fifteenth International Conference on Organic Synthesis (ICOS-15) (August 1-6, 2004, Nagoya, Japan), Prof. Minoru Isobe and Hisashi Yamamoto, ed. Organizng Committee of ICOS-15, International Union of Pure and Applied Chemistry (IUPAC)
Synthetic Studies on Cyathin Core
Fifteenth International Conference on Organic Synthesis (ICOS-15) (August 1-6, 2004, Nagoya, Japan), Prof. Minoru Isobe and Hisashi Yamamoto, ed. Organizng Committee of ICOS-15, International Union of Pure and Applied Chemistry (IUPAC)
First total synthesis of antimitotic compound, (+)-phomopsidin
The 229th ACS National Meeting (San Diego, CA, March 13-17, 2005)g Committee of ICOS-15, International Union of Pure and Applied Chemistry (IUPAC)
Synthetic Studies on Taxol
The 229th ACS National Meeting (San Diego, CA, March 13-17, 2005), The American Chemical Society, 559 (2005)
Synthetic studies on FR182877
The 229th ACS National Meeting (San Diego, CA, March 13-17, 2005), The American Chemical Society, 559 (2005)
Synthetic studies on Erinacines
The 229th ACS National Meeting (San Diego, CA, March 13-17, 2005), The American Chemical Society, 562 (2005)
FR182877の全合成研究(1)
日本化学会第85春季年会 神奈川
新規キラルシントンの創製と天然物合成への応用
日本化学会第85春季年会 神奈川
オフィオボリンAの全合成研究
日本化学会第85春季年会 神奈川
FR182877の全合成研究(2)
日本化学会第85春季年会 神奈川
(-)-Lepadiformineの不斉全合成研究
日本化学会第85春季年会 神奈川
触媒的不斉野崎-檜山反応による光学活性アレニルアルコールとホモプロパルギルアルコールの選択的合成
日本化学会第85春季年会 神奈川
(+)-digitoxigeninの合成研究
日本化学会第85春季年会 神奈川
抗腫瘍性化合物Taxolの不斉全合成研究(1)
日本化学会第85春季年会 神奈川
抗腫瘍性化合物Taxolの不斉全合成研究(2)
日本化学会第85春季年会 神奈川
(+)-アロサイアチンB2の不斉全合成
日本化学会第85春季年会 神奈川
(+)-phomopsidinの全合成
第85回有機合成シンポジウム
光学活性カルバゾール配位子を用いた触媒的不斉野崎ー檜山反応
第86回有機合成シンポジウム
触媒的不斉分子内シクロプロパン化反応の研究と天然物合成への応用展開
第48回有機合成化学協会関東支部シンポジウム
Erinacine 類の効率的不斉全合成研究
第30回反応と合成の進歩シンポジウム
erinacine 類の不斉全合成研究
日本薬学会125年会
分子内野崎-檜山反応、分子内鈴木-宮浦カップリングを用いたタキサン骨格の合成法研究
日本薬学会125年会
配位子及び不斉触媒
中田 雅久
Patent
2008 年度(第1回)有機合成化学協会 アステラス製薬・生命有機化学賞
2008 有機合成化学協会
日本薬学会奨励賞
1997
縮環部全炭素四級不斉中心の構築と異種生物活性多環式化合物の不斉全合成に関する研究
Project Year :
反応集積化が導く中分子戦略:高次生物機能分子の創製
Project Year :
Efficient Synthesis of Important Bioactive Medium-Size Polycyclic Natural Products
Project Year :
Research on Asymmetric Catalysis Based on Design and Synthesis of New Chiral Pincer-Type NHC Ligand
Project Year :
Catalytic Asymmetric Reactions of Alkenes Activated by Two Electron-Withdrawing Groups and Their Applications to Efficient Enantioselective Total Syntheses
Project Year :
Research on Asymmetric Catalysis Based on Design and Synthesis of New Chiral Pincer-Type NHC Ligand
Project Year :
2つの電子求引基で活性化されたアルケンの不斉触媒反応と効率的不斉全合成への活用
科学研究費助成事業(早稲田大学) 科学研究費助成事業(基盤研究(B))
Project Year :
Catalytic Asymmetric Reactions of Alkenes Activated by Two Electron-Withdrawing Groups and Their Applications to Efficient Enantioselective Total Syntheses
Project Year :
Organic Synthesis Based on Reaction Integration. Development of New Methods and Creation of New Substances
Project Year :
Synthetic Studies on Bioactive Natural Products utilizing Integrated
Project Year :
Research on the design and synthesis of chiral NHC pincer ligands and their utility for asymmetric catalysis
Project Year :
生理活性素材開発
文部科学省
Project Year :
Catalytic Asymmetric Synthesis of Bioactive Molecules with a Benzylic Quarternary Carbon
抗腫瘍性マクロリド、リゾキシンの構造活性相関及び生物有機化学的研究
プロティンナーゼC活性化調節機構の分子レベルで解明に関する研究
PI3キナーゼ阻害剤ワ-トマンニンの合成と生物有機化学的展開
Total Synthesis of Natural Products Possessing Multiple Bioactivities and Isolation of Their Activities
生合成類似ルートによる抗腫瘍性テルペノイド,タキソールの合成研究
Synthetic Study on Taxol via a New Route Inspired by Its Biogenesis
生物活性多環式天然物の効率的全合成研究
Studies on the total synthesis and SAR of natural products that bind to tublin
生物活性多環式天然物の効率的全合成研究
Preparation of new chiral building blocks and their practical use in the enantioselective total synthesis of bioactive polycyclic natural products
生体分子の一分子検出・機能解析システムの開発と応用
タキソールの不斉全合成研究
第93回有機合成シンポジウム
Presentation date: 2008.06
MK8383の不斉全合成
第55回有機合成化学協会関東シンポジウム
Presentation date: 2008.05
Studies on Enantioselective Total Syntehsis of (+)-Ophiobolin A
Presentation date: 2008.03
Taxolの収束的不斉全合成研究
日本薬学会第128年会
Presentation date: 2008.03
(+)-Ophiobolin Aの不斉全合成研究
日本化学会第88春季年会
Presentation date: 2008.03
Studies on Asymmetric Total Synthesis of
Presentation date: 2008.03
Synthetic Studies on (-)-FR182877(1)
Presentation date: 2008.03
Synthetic Studies on MK8383
Presentation date: 2008.03
Synthetic studies on (+)-bucidarasin C
Presentation date: 2008.03
Enantioselective Total Synthesis of (-)-Erinacine E
Presentation date: 2008.03
Studies on Convergent and Enantioselective Total Synthesis of Taxol
Presentation date: 2008.03
Biomimetic Total Synthesis of (−)-Erinacine E
9th Annual Florida Heterocyclic and Synthetic IUPAC-Sponsored Conference
Presentation date: 2008.03
Studies on Convergent and Enantioselective Total Synthesis of Taxol
9th Annual Florida Heterocyclic and Synthetic IUPAC-Sponsored Conference
Presentation date: 2008.03
Biomimetic Total Synthesis of (−)-Erinacine E
9th Annual Florida Heterocyclic and Synthetic IUPAC-Sponsored Conference
Presentation date: 2008.03
Synthetic Studies on (-)-FR182877(2)
Presentation date: 2008.02
First Enantioselective Total Synthesis of FR901512 via the Catalytic Asymmetric Nozaki-Hiyama Reactions
Catalysis & Fine Chemicals 2007 (C&FC 2007)
Presentation date: 2007.12
ハイパーフォリンの不斉全合成研究
第54回有機合成化学協会関東支部シンポジウム (新潟シンポジウム)
Presentation date: 2007.12
(+)-Phomopsidinの改良不斉全合成
第92回有機合成シンポジウム
Presentation date: 2007.11
Development of Catalytic Asymmetric Nozaki-Hiyama Reactions and their Application to Enantioselective Total Synthesis of FR901512
14th IUPAC International Symposium on Organometallic Chemistry Directed Towards Organic Synthesis (OMCOS 14)
Presentation date: 2007.08
(+)-ophiobolin Aの不斉全合成研究
第91回有機合成シンポジウム
Presentation date: 2007.06
Synthetic Studies on Polycyclic Polyprenylated Acylphloroglucinols
Presentation date: 2007.06
hyperforinの不斉全合成研究
第53回有機合成化学協会関東支部シンポジウム 横浜シンポジウム
Presentation date: 2007.05
Design of Catalytic Asymmetric Reactions and their Applications to Enantioselective Total Synthesis of Bioactive Natural Products
Molecular Chirality 2007 (MC 2007)
Presentation date: 2007.05
抗腫瘍性化合物Taxolの不斉全合成研究:エポキシドに対しての1,5-ヒドリドシフトによるtrans縮環したB,C環部位構築
日本薬学会第127年会
Presentation date: 2007.03
(+)-ophiobolin Aの不斉全合成研究
日本薬学会第127年会
Presentation date: 2007.03
エリナシンBの不斉全合成
日本薬学会第127年会
Presentation date: 2007.03
(-)-タキソールの不斉全合成研究
日本化学会第87春季年会
Presentation date: 2007.03
(-)-FR182877の全合成研究
日本化学会第87春季年会
Presentation date: 2007.03
(-)-physostigmineの形式全合成
日本化学会第87春季年会
Presentation date: 2007.03
ハイパーフォリンの不斉全合成研究
日本化学会第87春季年会
Presentation date: 2007.03
2017 Yuta Oki
不斉NHC配位子の開発に基づく不斉触媒反応創出と生物活性化合物の不斉全合成研究
2017 Yuta Oki
2014
2004
Special Laboratory on Chemistry and Biochemistry
Graduate School of Advanced Science and Engineering
2022 full year
Seminar on Chemical Synthesis Methods D
Graduate School of Advanced Science and Engineering
2022 fall semester
Seminar on Chemical Synthesis Methods C
Graduate School of Advanced Science and Engineering
2022 spring semester
Seminar on Chemical Synthesis Methods B
Graduate School of Advanced Science and Engineering
2022 fall semester
Seminar on Chemical Synthesis Methods A
Graduate School of Advanced Science and Engineering
2022 spring semester
Graduate School of Advanced Science and Engineering
2022 an intensive course(spring and fall)
Research on Chemical Synthesis Method
Graduate School of Advanced Science and Engineering
2022 full year
Master's Thesis (Department of Chemistry and Biochemistry)
Graduate School of Advanced Science and Engineering
2022 full year
Master's Thesis (Department of Chemistry and Biochemistry)
Graduate School of Advanced Science and Engineering
2022 full year
Seminar on Chemical Synthesis Methods D
Graduate School of Advanced Science and Engineering
2022 fall semester
Seminar on Chemical Synthesis Methods C
Graduate School of Advanced Science and Engineering
2022 spring semester
Seminar on Chemical Synthesis Methods B
Graduate School of Advanced Science and Engineering
2022 fall semester
Seminar on Chemical Synthesis Methods A
Graduate School of Advanced Science and Engineering
2022 spring semester
Experiments in Chemistry and Biochemistry
Graduate School of Advanced Science and Engineering
2022 full year
Research on Chemical Synthesis Method
Graduate School of Advanced Science and Engineering
2022 full year
Research on Chemical Synthesis Method
Graduate School of Advanced Science and Engineering
2022 full year
Special Seminar Abroad on Chemistry and Biochemistry
Graduate School of Advanced Science and Engineering
2022 full year
Special Seminar on Chemistry and Biochemistry B
Graduate School of Advanced Science and Engineering
2022 fall semester
Special Seminar on Chemistry and Biochemistry A
Graduate School of Advanced Science and Engineering
2022 spring semester
Science and Engineering Laboratory 1B V
School of Fundamental Science and Engineering
2022 fall semester
Science and Engineering Laboratory 1A III
School of Fundamental Science and Engineering
2022 spring semester
Science and Engineering Laboratory 1B V
School of Creative Science and Engineering
2022 fall semester
Science and Engineering Laboratory 1A III
School of Creative Science and Engineering
2022 spring semester
Science and Engineering Laboratory 1A III
School of Advanced Science and Engineering
2022 spring semester
Basic Experiments in Science and Engineering 2B Butsuri
School of Advanced Science and Engineering
2022 fall semester
Basic Experiments in Science and Engineering 2B Oubutsu
School of Advanced Science and Engineering
2022 fall semester
Science and Engineering Laboratory 1B V
School of Advanced Science and Engineering
2022 fall semester
Organic Chemistry : Experiment [S Grade]
School of Advanced Science and Engineering
2022 spring semester
Organic Chemistry : Exercises [S Grade]
School of Advanced Science and Engineering
2022 fall semester
Organic Chemistry Laboratory [S Grade]
School of Advanced Science and Engineering
2022 fall semester